Key Takeaways

  • Respiratory depression is the most serious opioid adverse effect - assess respiratory rate before EVERY dose; hold if RR < 12/min
  • Naloxone (Narcan) is the antidote for opioid overdose - it has a shorter half-life than most opioids, so re-sedation can occur
  • Opioid-naive patients are at highest risk for respiratory depression - start low and titrate slowly
  • Constipation is an expected side effect that does NOT develop tolerance - prophylactic bowel regimen is essential
  • Assess pain using validated scales; do not rely solely on vital signs or patient appearance
Last updated: January 2026

High-Alert Medications: Opioids

Opioid analgesics are essential for pain management but carry significant risks. The NCLEX tests your ability to safely administer opioids, recognize adverse effects, and respond to emergencies.

Common Opioid Analgesics

DrugRouteRelative PotencyDuration
MorphinePO, IV, IM, SubQStandard (1x)4-5 hours
Hydromorphone (Dilaudid)PO, IV5-7x morphine4-5 hours
FentanylIV, Transdermal, Transmucosal80-100x morphineIV: 30-60 min; Patch: 72 hr
OxycodonePO1.5x morphine4-6 hours
HydrocodonePO~1x morphine4-6 hours
CodeinePO0.1x morphine4-6 hours
Meperidine (Demerol)PO, IM0.1x morphine2-3 hours

Clinical Note: Meperidine is rarely used due to neurotoxic metabolite (normeperidine) that can cause seizures.

Before Administration: The Opioid Assessment

ALWAYS assess before each dose:

  1. Respiratory Rate - Hold if < 12 breaths/min
  2. Level of Consciousness - Excessive sedation = hold and assess
  3. Pain Score - Document current pain level
  4. Last Dose Time - Verify minimum interval has passed
  5. Allergies - True allergy vs. expected side effect
  6. Other CNS Depressants - Benzodiazepines, alcohol increase risk

Respiratory Depression: The Priority Concern

Signs of Opioid-Induced Respiratory Depression:

  • Respiratory rate < 12/min
  • Shallow respirations
  • Oxygen saturation declining
  • Excessive sedation (difficult to arouse)
  • Snoring or obstructed breathing

Sedation Scale (Pasero Opioid-Induced Sedation Scale):

LevelDescriptionAction
S = SleepNormal sleep, easily arousedNone
1Awake and alertNone
2Slightly drowsy, easily arousedAcceptable
3Frequently drowsy, arousableDecrease dose; monitor closely
4Somnolent, minimal responseStop opioid; call provider; consider Naloxone

Naloxone (Narcan): Opioid Reversal

Indications:

  • Respiratory depression (RR < 8-10/min)
  • Unresponsive to stimulation
  • Oxygen saturation falling despite supplemental O2

Administration:

  • IV: 0.4-2 mg every 2-3 minutes until response
  • IM, SubQ, or Intranasal if no IV access
  • Titrate to respiratory improvement, NOT complete reversal

Critical Concept: Naloxone has a shorter half-life (30-90 min) than most opioids (4-5 hours). Re-sedation can occur. Monitor for at least 2 hours after administration; may need repeat doses.

Side Effects of Rapid Reversal:

  • Severe pain return
  • Hypertension, tachycardia
  • Pulmonary edema
  • Withdrawal symptoms in opioid-dependent patients

Managing Opioid Side Effects

Side EffectManagement
ConstipationProphylactic stool softener + stimulant laxative (does NOT develop tolerance)
Nausea/VomitingAntiemetics; usually improves after 2-3 days
Pruritus (itching)Antihistamines; not a true allergy
Urinary retentionBladder assessment; may need catheterization
HypotensionSlow position changes; assess fluid status
SedationExpected initially; assess for excessive sedation

Opioid-Naive vs. Opioid-Tolerant

Opioid-NaiveOpioid-Tolerant
No recent opioid useRegular opioid use > 1 week
Higher risk of respiratory depressionMay need higher doses for effect
Start with lower dosesCross-tolerance to other opioids
Titrate slowlyStill at risk if doses increased

Equianalgesic Dosing

When converting between opioids, use equianalgesic charts:

OpioidOral DoseIV Dose
Morphine30 mg10 mg
Hydromorphone6 mg1.5 mg
Oxycodone20 mgN/A

Remember: These are approximations. Incomplete cross-tolerance means starting 25-50% below calculated dose.

Patient-Controlled Analgesia (PCA)

Safety Features:

  • Lockout interval prevents overdose
  • Basal rate (if ordered) provides continuous relief
  • Patient activates demand doses
  • Only the PATIENT should push the button (not family)

Nursing Responsibilities:

  • Verify pump settings with two nurses
  • Assess pain and sedation regularly
  • Document usage and pain scores
  • Teach patient proper use

Special Populations

Elderly:

  • Start at 25-50% of usual adult dose
  • Longer duration of action (slower metabolism)
  • Higher risk of falls, confusion

Renal Impairment:

  • Morphine metabolites accumulate - consider alternatives
  • Hydromorphone or fentanyl often preferred

Hepatic Impairment:

  • Reduced metabolism - lower doses needed
  • Extended duration of action

On the Exam

  • Respiratory assessment before every opioid dose
  • Know when to hold medication (RR < 12)
  • Recognize need for Naloxone
  • Understand that constipation requires prophylaxis
  • PCA - only patient pushes button
Test Your Knowledge

A patient receiving IV morphine has a respiratory rate of 8/min, is difficult to arouse, and has oxygen saturation of 88%. The nurse's priority action is:

A
B
C
D
Test Your Knowledge

After administering Naloxone for opioid overdose, the nurse should:

A
B
C
D
Test Your Knowledge

Which opioid side effect does NOT develop tolerance over time?

A
B
C
D
Test Your Knowledge

A patient with a PCA pump appears over-sedated. The family member states, "I've been pushing the button for him so he can rest." The nurse should:

A
B
C
D